Brief Information of the Compound and Protein
Compound Name
Rac-2'-chloro-N-((2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl)-6-((2,3-dihydrobenzofuran-6-yl)methylamino)-3,4'-bipyridine-5-carboxamide
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PubChem ID
CID: 122180021
Canonical SMILES
O=C(NCC1COc2ccccc2O1)c1cc(-c2ccnc(Cl)c2)cnc1NCc1ccc2c(c1)OCC2
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Compound Formula C29H25ClN4O4
Compound Structure
Protein Name
Growth hormone secretagogue receptor type 1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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GRP-related receptor
Uniprot ID
O08725
Gene Name
GHSR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 390 nM
   TI
   LI
   LO
   TS