Brief Information of the Compound and Protein
Compound Name
(R)-4-((9-Chloro-7-(5-fluoro-1H-indol-1-yl)-3-methyl-2,3-dihydrobenzo[f][1,4]oxazepin-4(5H)-yl)methyl)pyridin-2(1H)-one
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PubChem ID
CID: 122180297
Canonical SMILES
C[C@@H]1COc2c(Cl)cc(-n3ccc4cc(F)ccc43)cc2CN1Cc1cc[nH]c(=O)c1
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Compound Formula C24H21ClFN3O2
Compound Structure
Protein Name
Prostaglandin E2 receptor EP1 subtype
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Lipid-like ligand receptor (family A GPCR)
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Prostanoid receptor
Uniprot ID
P34995
Gene Name
PTGER1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000516 ECV-304 Homo sapiens (Human)  1
1
IC50 > 30000 nM
   TI
   LI
   LO
   TS