Brief Information of the Compound and Protein
Compound Name
 Compound Info 
2,2,4,4-Tetramethyl-6-(pyrazolo[1,5-a]pyridin-4-yl)-2,3,4,7,8,9-hexahydro-1H-cyclopenta[h]quinolin-3-one
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 PubChem ID
CID: 59233334
Canonical SMILES
CC1(C)Nc2c(cc(-c3cccn4nccc34)c3c2CCC3)C(C)(C)C1=O
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Compound Formula C23H25N3O
Compound Structure
Protein Name
 Protein Info 
Glucocorticoid receptor
Protein Classification
Transcription factor
>
Nuclear receptor
>
Nuclear hormone receptor subfamily 3
>
Nuclear hormone receptor subfamily 3 group C
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Nuclear hormone receptor subfamily 3 group C member 1
Uniprot ID
P04150
Gene Name
NR3C1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
IC50 = 84 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 Ki = 35 nM