Brief Information of the Compound and Protein
Compound Name
2-(benzylamino)-6-(1H-pyrazole-5-carbonyl)-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carbonitrile
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PubChem ID
CID: 118735959
Canonical SMILES
O=C(N1CCc2c(C1)sc(NCc1ccccc1)c2C#N)c1ccn[nH]1
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Compound Formula C19H17N5OS
Compound Structure
Protein Name
Metabotropic glutamate receptor 1
Protein Classification
Membrane receptor
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Family C G protein-coupled receptor
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Small molecule receptor (family C GPCR)
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Neurotransmitter receptor (family C GPCR)
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Metabotropic glutamate receptor
Uniprot ID
Q13255
Gene Name
GRM1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000447 Chem-3 Mus musculus (Mouse)  1
1
IC50 = 1090 nM
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