Brief Information of the Compound and Protein
Compound Name
 Compound Info 
(5-bromo-1-methylpyrrolo[2,3-c]pyridin-2-yl)-[6-[(dimethylamino)methyl]-3,4-dihydro-1H-isoquinolin-2-yl]methanone
    Show/Hide
 PubChem ID
CID: 118707553
Canonical SMILES
CN(C)Cc1ccc2CN(CCc2c1)C(=O)c1cc2cc(Br)ncc2n1C
    Show/Hide
Compound Formula C21H23BrN4O
Compound Structure
Protein Name
 Protein Info 
Pyroglutamylated RF-amide peptide receptor
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Peptide receptor (family A GPCR)
>
Short peptide receptor (family A GPCR)
>
RF amide receptor
Uniprot ID
Q96P65
Gene Name
QRFPR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
IC50 = 240 nM
   TI
   LI
   LO
   TS
CL000006 HEK293
 Cell Line Info 
Homo sapiens (Human)  1
1
IC50 = 280 nM
   TI
   LI
   LO
   TS