Brief Information of the Compound and Protein
Compound Name
 Compound Info 
(10R,15S)-12-[3-(6-fluoro-2H-indazol-3-yl)propyl]-4-methyl-1,4,12-triazatetracyclo[7.6.1.05,16.010,15]hexadeca-5,7,9(16)-triene
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 PubChem ID
CID: 90655118
Canonical SMILES
CN1CCN2[C@H]3CCN(CCCc4n[nH]c5cc(F)ccc45)C[C@H]3c3cccc1c23
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Compound Formula C24H28FN5
Compound Structure
Protein Name
 Protein Info 
5-hydroxytryptamine receptor 2A
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Serotonin receptor
Uniprot ID
P28223
Gene Name
HTR2A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000065 HEK293-EBNA
 Cell Line Info 
Homo sapiens (Human)  1
1
Ki = 18 nM
   TI
   LI
   LO
   TS