Brief Information of the Compound and Protein
Compound Name
4-[4-(4-Cyano-3-fuoro-phenoxymethyl)-4-hydroxy-piperidine-1-sulfonyl]-isophthalonitrile
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PubChem ID
CID: 90665453
Canonical SMILES
N#Cc1ccc(S(=O)(=O)N2CCC(O)(COc3ccc(C#N)c(F)c3)CC2)c(C#N)c1
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Compound Formula C21H17FN4O4S
Compound Structure
Protein Name
Transient receptor potential cation channel subfamily V member 4
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q9HBA0
Gene Name
TRPV4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  1
1
IC50 = 50.5 nM
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