Brief Information of the Compound and Protein
Compound Name
2-(4-phenoxyphenyl)-1-[2-(trifluoromethyl)-5,11-dihydropyrido[3,2-c][1,5]benzodiazepin-6-yl]ethanone
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PubChem ID
CID: 76314246
Canonical SMILES
FC(F)(F)c1ccc2CN(C(=O)Cc3ccc(Oc4ccccc4)cc3)c3ccccc3Nc2n1
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Compound Formula C27H20F3N3O2
Compound Structure
Protein Name
Bombesin receptor subtype-3
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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GRP-related receptor
Uniprot ID
P32247
Gene Name
BRS3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  1
1
EC50 = 368 nM
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