Brief Information of the Compound and Protein
Compound Name
 Compound Info 
2-(4-tert-butylphenyl)-1-[2-(trifluoromethyl)-5,11-dihydropyrido[3,2-c][1,5]benzodiazepin-6-yl]ethanone
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 PubChem ID
CID: 76317822
Canonical SMILES
CC(C)(C)c1ccc(CC(=O)N2Cc3ccc(nc3Nc3ccccc23)C(F)(F)F)cc1
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Compound Formula C25H24F3N3O
Compound Structure
Protein Name
 Protein Info 
Bombesin receptor subtype-3
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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GRP-related receptor
Uniprot ID
O54798
Gene Name
BRS3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
EC50 = 227 nM
   TI
   LI
   LO
   TS