Brief Information of the Compound and Protein
Compound Name
5-(3-cyclobutyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yloxy)-N-methylpyrazine-2-carboxamide
    Show/Hide
PubChem ID
CID: 10473209
SID: 15496737
Canonical SMILES
CNC(=O)c1cnc(Oc2ccc3CCN(CCc3c2)C2CCC2)cn1
    Show/Hide
Compound Formula C20H24N4O2
Compound Structure
Protein Name
Histamine H3 receptor
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Small molecule receptor (family A GPCR)
>
Monoamine receptor
>
Histamine receptor
Uniprot ID
Q9QYN8
Gene Name
HRH3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Ki = 1.122 nM
   TI
   LI
   LO
   TS