Brief Information of the Compound and Protein
Compound Name
4'-((4-((3,4-Dihydro-2H-[1,3]oxazino[3,2-a]indole-10-carboxamido)methyl)piperidin-1-yl)methyl)[1,1'-biphenyl]-2-carboxylic acid
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PubChem ID
CID: 72697441
Canonical SMILES
O=C(O)c1ccccc1-c1ccc(CN2CCC(CNC(=O)c3c4n(c5ccccc35)CCCO4)CC2)cc1
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Compound Formula C32H33N3O4
Compound Structure
Protein Name
5-hydroxytryptamine receptor 4
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Serotonin receptor
Uniprot ID
Q13639
Gene Name
HTR4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Ki = 0.631 nM
   TI
   LI
   LO
   TS