Brief Information of the Compound and Protein
Compound Name
3-[1-(4-fluorophenyl)indazol-5-yl]-2,2-dimethyl-3-phenyl-N-(triazol-2-yl)propanamide
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PubChem ID
CID: 73346225
Canonical SMILES
CC(C)(C(c1ccccc1)c1ccc2n(ncc2c1)-c1ccc(F)cc1)C(=O)Nn1nccn1
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Compound Formula C26H23FN6O
Compound Structure
Protein Name
Glucocorticoid receptor
Protein Classification
Transcription factor
>
Nuclear receptor
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Nuclear hormone receptor subfamily 3
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Nuclear hormone receptor subfamily 3 group C
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Nuclear hormone receptor subfamily 3 group C member 1
Uniprot ID
P04150
Gene Name
NR3C1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000068 A-549 Homo sapiens (Human)  1
1
EC50 = 17 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 Ki = 11 nM