Brief Information of the Compound and Protein
Compound Name
methyl 2-[4-[4-[5,6-dichloro-4-(dimethylcarbamoyl)-2-(propan-2-ylamino)benzimidazol-1-yl]piperidin-1-yl]phenyl]-2-methylpropanoate
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PubChem ID
CID: 71528732
SID: 163522082
Canonical SMILES
COC(=O)C(C)(C)c1ccc(cc1)N1CCC(CC1)n1c(NC(C)C)nc2c(C(=O)N(C)C)c(Cl)c(Cl)cc12
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Compound Formula C29H37Cl2N5O3
Compound Structure
Protein Name
Transient receptor potential cation channel subfamily V member 4
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q9HBA0
Gene Name
TRPV4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 15.8 nM
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