Brief Information of the Compound and Protein
Compound Name
5,6-dichloro-1-[1-(4-chlorophenyl)sulfonylpiperidin-4-yl]-N,N-dimethyl-2-(propan-2-ylamino)benzimidazole-4-carboxamide
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PubChem ID
CID: 71528448
SID: 163521782
Canonical SMILES
CC(C)Nc1nc2c(C(=O)N(C)C)c(Cl)c(Cl)cc2n1C1CCN(CC1)S(=O)(=O)c1ccc(Cl)cc1
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Compound Formula C24H28Cl3N5O3S
Compound Structure
Protein Name
Transient receptor potential cation channel subfamily V member 4
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q9HBA0
Gene Name
TRPV4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 3980 nM
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