Brief Information of the Compound and Protein
Compound Name
rac-4-(Biphenyl-4-yl)-N-(4-methoxybenzyl)-2,7,7-trimethyl-5-oxo-1,4,5,6,7,8-hexahydroquinoline-3-carboxamide
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PubChem ID
CID: 71459206
SID: 163502793
Canonical SMILES
COc1ccc(CNC(=O)C2=C(C)NC3=C(C(=O)CC(C)(C)C3)C2c2ccc(-c3ccccc3)cc2)cc1
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Compound Formula C33H34N2O3
Compound Structure
Protein Name
TGF-beta receptor type-2
Protein Classification
Enzyme
>
Kinase
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Protein Kinase
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TKL protein kinase group
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TKL protein kinase STKR family
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TKL protein kinase STKR Type 2 subfamily
Uniprot ID
P37173
Gene Name
TGFBR2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000025 HEK-293T Homo sapiens (Human)  1
1
IC50 = 4060 nM
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