Brief Information of the Compound and Protein
Compound Name
rac-Methyl 4-(Biphenyl-4-yl)-7-(4-(dimethylamino)phenyl)-2-methyl-5-oxo-1,4,5,6,7,8-hexahydroquinoline-3-carboxylate
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PubChem ID
CID: 71043140
SID: 163503152
Canonical SMILES
COC(=O)C1=C(C)NC2=C(C(=O)CC(c3ccc(N(C)C)cc3)C2)C1c1ccc(-c2ccccc2)cc1
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Compound Formula C32H32N2O3
Compound Structure
Protein Name
TGF-beta receptor type-2
Protein Classification
Enzyme
>
Kinase
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Protein Kinase
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TKL protein kinase group
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TKL protein kinase STKR family
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TKL protein kinase STKR Type 2 subfamily
Uniprot ID
P37173
Gene Name
TGFBR2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000025 HEK-293T Homo sapiens (Human)  1
1
IC50 = 3970 nM
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