Brief Information of the Compound and Protein
Compound Name
rac-Methyl 2,7,7-Trimethyl-5-oxo-4-(4'-(trifluoromethyl)biphenyl-4-yl)-1,4,5,6,7,8-hexahydroquinoline-3-carboxylate
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PubChem ID
CID: 71453843
SID: 163503511
Canonical SMILES
COC(=O)C1=C(C)NC2=C(C(=O)CC(C)(C)C2)C1c1ccc(-c2ccc(C(F)(F)F)cc2)cc1
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Compound Formula C27H26F3NO3
Compound Structure
Protein Name
TGF-beta receptor type-2
Protein Classification
Enzyme
>
Kinase
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Protein Kinase
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TKL protein kinase group
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TKL protein kinase STKR family
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TKL protein kinase STKR Type 2 subfamily
Uniprot ID
P37173
Gene Name
TGFBR2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000025 HEK-293T Homo sapiens (Human)  1
1
IC50 = 730 nM
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