Brief Information of the Compound and Protein
Compound Name
3-[2,6-dimethoxy-4-(methoxymethyl)phenyl]-6-methoxy-N-(oxan-4-yl)-N-propan-2-ylpyrazolo[5,1-b][1,3]thiazol-7-amine
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PubChem ID
CID: 71453735
SID: 163490916
Canonical SMILES
COCc1cc(OC)c(-c2csc3c(N(C(C)C)C4CCOCC4)c(OC)nn23)c(OC)c1
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Compound Formula C24H33N3O5S
Compound Structure
Protein Name
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
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Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Corticotropin releasing factor receptor
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Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 136 nM
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