Brief Information of the Compound and Protein
Compound Name
3,5-dimethoxy-4-[6-methoxy-7-[oxan-4-yl(propyl)amino]pyrazolo[5,1-b][1,3]thiazol-3-yl]benzonitrile
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PubChem ID
CID: 71459110
SID: 163490919
Canonical SMILES
CCCN(C1CCOCC1)c1c(OC)nn2c(csc12)-c1c(OC)cc(cc1OC)C#N
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Compound Formula C23H28N4O4S
Compound Structure
Protein Name
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
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Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Corticotropin releasing factor receptor
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Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 126 nM
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