Brief Information of the Compound and Protein
Compound Name
4-fluoro-6-[(1-propylpiperidin-4-yl)methoxy]phenanthridine
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PubChem ID
CID: 71461050
SID: 163506329
Canonical SMILES
CCCN1CCC(COc2nc3c(F)cccc3c3ccccc23)CC1
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Compound Formula C22H25FN2O
Compound Structure
Protein Name
5-hydroxytryptamine receptor 4
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Serotonin receptor
Uniprot ID
Q13639
Gene Name
HTR4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000025 HEK-293T Homo sapiens (Human)  2
1
EC50 = 63.1 nM
   TI
   LI
   LO
   TS
2
Ki = 3.1 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 Ki = 3.1 nM