Brief Information of the Compound and Protein
Compound Name
4-methoxy-6-[(1-propylpiperidin-4-yl)methoxy]phenanthridine
    Show/Hide
PubChem ID
CID: 71461049
SID: 163505986
Canonical SMILES
CCCN1CCC(COc2nc3c(OC)cccc3c3ccccc23)CC1
    Show/Hide
Compound Formula C23H28N2O2
Compound Structure
Protein Name
5-hydroxytryptamine receptor 4
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Small molecule receptor (family A GPCR)
>
Monoamine receptor
>
Serotonin receptor
Uniprot ID
Q13639
Gene Name
HTR4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000025 HEK-293T Homo sapiens (Human)  2
1
EC50 = 79.4 nM
   TI
   LI
   LO
   TS
2
Ki = 17 nM
   TI
   LI
   LO
   TS