Brief Information of the Compound and Protein
Compound Name
 Compound Info 
rac-2-(3-Fluoro-4-(methylsulfonamido)phenyl)-N-((2-(piperidin-1-yl)-6-(trifluoromethyl)pyridin-3-yl)methyl)propanamide
    Show/Hide
 PubChem ID
CID: 16223604
SID: 24906077
Canonical SMILES
CC(C(=O)NCc1ccc(C(F)(F)F)nc1N1CCCCC1)c1ccc(NS(C)(=O)=O)c(F)c1
    Show/Hide
Compound Formula C22H26F4N4O3S
Compound Structure
Protein Name
 Protein Info 
Transient receptor potential cation channel subfamily V member 1
Protein Classification
Ion channel
>
Voltage-gated ion channel
>
Transient receptor potential channel
Uniprot ID
Q8NER1
Gene Name
TRPV1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  2
1
IC50 = 218 nM
   TI
   LI
   LO
   TS
2
Ki = 0.43 nM
   TI
   LI
   LO
   TS