Brief Information of the Compound and Protein
Compound Name
 Compound Info 
2-[3-fluoro-4-(methanesulfonamido)phenyl]-N-[[2-(4-pyridin-2-ylpiperazin-1-yl)-6-(trifluoromethyl)pyridin-3-yl]methyl]propanamide
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 PubChem ID
CID: 67439554
SID: 163489339
Canonical SMILES
CC(C(=O)NCc1ccc(nc1N1CCN(CC1)c1ccccn1)C(F)(F)F)c1ccc(NS(C)(=O)=O)c(F)c1
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Compound Formula C26H28F4N6O3S
Compound Structure
Protein Name
 Protein Info 
Transient receptor potential cation channel subfamily V member 1
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q8NER1
Gene Name
TRPV1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  2
1
IC50 = 108 nM
   TI
   LI
   LO
   TS
2
Ki = 1.4 nM
   TI
   LI
   LO
   TS