Brief Information of the Compound and Protein
Compound Name
 Compound Info 
[3-[6-(4-tert-butylphenyl)sulfonyl-2-(trifluoromethyl)-5,11-dihydropyrido[3,2-c][1,5]benzodiazepin-7-yl]-1,2,4-oxadiazol-5-yl]methanol
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 PubChem ID
CID: 59618753
SID: 148139026
Canonical SMILES
CC(C)(C)c1ccc(cc1)S(=O)(=O)N1Cc2ccc(nc2Nc2cccc(-c3noc(CO)n3)c12)C(F)(F)F
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Compound Formula C26H24F3N5O4S
Compound Structure
Protein Name
 Protein Info 
Bombesin receptor subtype-3
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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GRP-related receptor
Uniprot ID
O54798
Gene Name
BRS3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000866 HEK293 AequoScreen
 Cell Line Info 
Homo sapiens (Human)  1
1
EC50 = 93 nM
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   LI
   LO
   TS