Brief Information of the Compound and Protein
Compound Name
2-[2,6-dimethoxy-4-(methoxymethyl)phenyl]-N-ethyl-8-methoxy-N-(2-methoxyethyl)-3-methylquinolin-5-amine
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PubChem ID
CID: 71451516
SID: 163447729
Canonical SMILES
CCN(CCOC)c1ccc(OC)c2nc(c(C)cc12)-c1c(OC)cc(COC)cc1OC
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Compound Formula C26H34N2O5
Compound Structure
Protein Name
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
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Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Corticotropin releasing factor receptor
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Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 392 nM
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