Brief Information of the Compound and Protein
Compound Name
[4-[3-[cyclopropylmethyl(oxan-4-ylmethyl)amino]-2-ethylpyrazolo[1,5-a]pyridin-7-yl]-3,5-dimethoxyphenyl]methanol
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PubChem ID
CID: 21084107
SID: 58104235
Canonical SMILES
CCc1nn2c(cccc2c1N(CC1CC1)CC1CCOCC1)-c1c(OC)cc(CO)cc1OC
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Compound Formula C28H37N3O4
Compound Structure
Protein Name
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
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Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Corticotropin releasing factor receptor
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Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 200 nM
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   LI
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