Brief Information of the Compound and Protein
Compound Name
 Compound Info 
2-[2,6-dimethoxy-4-(methoxymethyl)phenyl]-N,N-diethyl-3-fluoro-8-methylquinolin-5-amine
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 PubChem ID
CID: 70686533
SID: 163451566
Canonical SMILES
CCN(CC)c1ccc(C)c2nc(c(F)cc12)-c1c(OC)cc(COC)cc1OC
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Compound Formula C24H29FN2O3
Compound Structure
Protein Name
 Protein Info 
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
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Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Corticotropin releasing factor receptor
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Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293
 Cell Line Info 
Homo sapiens (Human)  2
1
IC50 = 131 nM
   TI
   LI
   LO
   TS
2
IC50 = 144 nM
   TI
   LI
   LO
   TS