Brief Information of the Compound and Protein
Compound Name
3-methyl-5-N,5-N-dipropyl-2-N-(2,4,6-trimethylphenyl)quinoxaline-2,5-diamine
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PubChem ID
CID: 70692630
SID: 163441221
Canonical SMILES
CCCN(CCC)c1cccc2nc(Nc3c(C)cc(C)cc3C)c(C)nc12
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Compound Formula C24H32N4
Compound Structure
Protein Name
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
>
Family B G protein-coupled receptor
>
Peptide receptor (family B GPCR)
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Corticotropin releasing factor receptor
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Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  2
1
IC50 = 155 nM
   TI
   LI
   LO
   TS
2
IC50 = 563 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 155 nM
2 IC50 = 563 nM