Brief Information of the Compound and Protein
Compound Name
2-[2,6-dimethoxy-4-(methoxymethyl)phenoxy]-N,N-diethyl-3-methylquinolin-5-amine
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PubChem ID
CID: 60141295
SID: 143484206
Canonical SMILES
CCN(CC)c1cccc2nc(Oc3c(OC)cc(COC)cc3OC)c(C)cc12
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Compound Formula C24H30N2O4
Compound Structure
Protein Name
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
>
Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Corticotropin releasing factor receptor
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Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  2
1
IC50 = 70 nM
   TI
   LI
   LO
   TS
2
IC50 = 167 nM
   TI
   LI
   LO
   TS