Brief Information of the Compound and Protein
Compound Name
 Compound Info 
2-(4-methoxy-2-methylphenyl)-7-methyl-5-pentan-3-yl-3H-pyrrolo[2,1-f][1,2,4]triazin-4-one
    Show/Hide
 PubChem ID
CID: 136042277
Canonical SMILES
CCC(CC)c1cc(C)n2nc([nH]c(=O)c12)-c1ccc(OC)cc1C
    Show/Hide
Compound Formula C20H25N3O2
Compound Structure
Protein Name
 Protein Info 
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
>
Family B G protein-coupled receptor
>
Peptide receptor (family B GPCR)
>
Corticotropin releasing factor receptor
>
Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  2
1
EC50 = 688 nM
   TI
   LI
   LO
   TS
2
IC50 = 149 nM
   TI
   LI
   LO
   TS