Brief Information of the Compound and Protein
Compound Name
(4aR,11R,11aS)-11-methyl-2-(2-piperidin-1-ylethyl)-9-(trifluoromethyl)-1,3,4,4a,5,6,11,11a-octahydropyrido[4,3-b]carbazole
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PubChem ID
CID: 57395050
Canonical SMILES
C[C@@H]1[C@H]2CN(CCN3CCCCC3)CC[C@@H]2Cc2[nH]c3ccc(cc3c12)C(F)(F)F
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Compound Formula C24H32F3N3
Compound Structure
Protein Name
Melanin-concentrating hormone receptor 1
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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MCH receptor
Uniprot ID
Q99705
Gene Name
MCHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000001 Jurkat Homo sapiens (Human)  1
1
IC50 = 100 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 40 nM