Brief Information of the Compound and Protein
Compound Name
4-[2-[(4aS,11S,11aR)-11-methyl-9-(trifluoromethyl)-1,3,4,4a,5,6,11,11a-octahydropyrido[4,3-b]carbazol-2-yl]ethyl]morpholine
    Show/Hide
PubChem ID
CID: 10202381
SID: 15200512
Canonical SMILES
C[C@H]1[C@@H]2CN(CCN3CCOCC3)CC[C@H]2Cc2[nH]c3ccc(cc3c12)C(F)(F)F
    Show/Hide
Compound Formula C23H30F3N3O
Compound Structure
Protein Name
Melanin-concentrating hormone receptor 1
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Peptide receptor (family A GPCR)
>
Short peptide receptor (family A GPCR)
>
MCH receptor
Uniprot ID
Q99705
Gene Name
MCHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000001 Jurkat Homo sapiens (Human)  1
1
IC50 = 1000 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 750 nM