Brief Information of the Compound and Protein
| Compound Name |
(1S,9R,13E)-1-amino-13-ethylidene-11-methyl-6-azatricyclo[7.3.1.02,7]trideca-2(7),3,10-trien-5-one
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PubChem ID | |||||
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Compound Structure |
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| Protein Name |
Acetylcholinesterase
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Protein Classification |
Enzyme
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Hydrolase
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| Uniprot ID | Gene Name | ACHE |
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Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
| Cell Line ID | Cell Line Name | Cell Line Organism | |
| CL000006 | HEK293 | Homo sapiens (Human) | 1 |
| 1 |
IC50 = 29 nM
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TI
LI
LO
TS
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|---|---|---|---|
Biochemical Assays
| 1 | IC50 = 0.54 nM | ||
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| 2 | IC50 = 5 nM | ||
| 3 | IC50 = 12 nM | ||
| 4 | IC50 = 21 nM | ||
| 5 | IC50 = 45 nM | ||
| 6 | IC50 = 47 nM | ||
| 7 | IC50 = 125 nM | ||
| 8 | IC50 = 150 nM | ||
| 9 | IC50 = 260 nM | ||
| 10 | IC50 = 1700 nM | ||
| 11 | Ki = 47 nM | ||