Brief Information of the Compound and Protein
Compound Name
 Compound Info 
4-[5-(2-morpholin-4-ylethoxy)pyridin-3-yl]-5,13,16-triazatetracyclo[8.6.0.02,7.011,15]hexadeca-1(10),2,4,6,8,11(15)-hexaen-12-one
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 PubChem ID
CID: 25066206
SID: 56403068
Canonical SMILES
O=C1NCc2[nH]c3c(ccc4cnc(cc34)-c3cncc(OCCN4CCOCC4)c3)c12
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Compound Formula C24H23N5O3
Compound Structure
Protein Name
 Protein Info 
MAP kinase-activated protein kinase 2
Protein Classification
Enzyme
>
Kinase
>
Protein Kinase
>
CAMK protein kinase group
>
CAMK protein kinase MAPKAPK family
>
CAMK protein kinase MAPKAPK subfamily
Uniprot ID
P49137
Gene Name
MAPKAPK2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000040 THP-1
 Cell Line Info 
Homo sapiens (Human)  1
1
IC50 = 9330 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 5 nM