Brief Information of the Compound and Protein
Compound Name
 Compound Info 
3-(benzenesulfonyl)-N,5,7-trimethylpyrazolo[1,5-a]pyrimidin-2-amine
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 PubChem ID
CID: 44516817
SID: 85851631
Canonical SMILES
CNc1nn2c(C)cc(C)nc2c1S(=O)(=O)c1ccccc1
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Compound Formula C15H16N4O2S
Compound Structure
Protein Name
 Protein Info 
5-hydroxytryptamine receptor 2B
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Serotonin receptor
Uniprot ID
P41595
Gene Name
HTR2B
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293
 Cell Line Info 
Homo sapiens (Human)  1
1
Ki = 1040 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 5130 nM