Brief Information of the Compound and Protein
Compound Name
 Compound Info 
2-[4-(1H-pyrazol-1-yl)phenyl]-1-(4-{[1-(trifluoromethyl)cyclopropyl]methyl}-1H-imidazol-2-yl)propan-2-ol
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 PubChem ID
CID: 25026044
SID: 56376707
Canonical SMILES
CC(O)(Cc1ncc(CC2(CC2)C(F)(F)F)[nH]1)c1ccc(cc1)-n1cccn1
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Compound Formula C20H21F3N4O
Compound Structure
Protein Name
 Protein Info 
Bombesin receptor subtype-3
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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GRP-related receptor
Uniprot ID
P32247
Gene Name
BRS3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000866 HEK293 AequoScreen
 Cell Line Info 
Homo sapiens (Human)  1
1
EC50 = 14 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 11 nM