Brief Information of the Compound and Protein
Compound Name
 Compound Info 
N-[(2S)-1-[[1-[3-[3-(hydroxymethyl)piperidine-1-carbonyl]phenyl]-6-methylindazol-4-yl]amino]propan-2-yl]cyclopropanesulfonamide
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 PubChem ID
CID: 53318326
Canonical SMILES
C[C@@H](CNc1cc(C)cc2n(ncc12)-c1cccc(c1)C(=O)N1CCCC(CO)C1)NS(=O)(=O)C1CC1
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Compound Formula C27H35N5O4S
Compound Structure
Protein Name
 Protein Info 
Glucocorticoid receptor
Protein Classification
Transcription factor
>
Nuclear receptor
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Nuclear hormone receptor subfamily 3
>
Nuclear hormone receptor subfamily 3 group C
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Nuclear hormone receptor subfamily 3 group C member 1
Uniprot ID
P04150
Gene Name
NR3C1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000068 A-549
 Cell Line Info 
Homo sapiens (Human)  2
1
IC50 = 251.19 nM
   TI
   LI
   LO
   TS
2
IC50 > 6309.57 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 125.89 nM