Brief Information of the Compound and Protein
Compound Name
 Compound Info 
N-[(2R)-2-[[1-(4-fluorophenyl)-6-methylindazol-4-yl]amino]propyl]-2,4,6-trimethylbenzenesulfonamide
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 PubChem ID
CID: 53321440
Canonical SMILES
C[C@H](CNS(=O)(=O)c1c(C)cc(C)cc1C)Nc1cc(C)cc2n(ncc12)-c1ccc(F)cc1
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Compound Formula C26H29FN4O2S
Compound Structure
Protein Name
 Protein Info 
Glucocorticoid receptor
Protein Classification
Transcription factor
>
Nuclear receptor
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Nuclear hormone receptor subfamily 3
>
Nuclear hormone receptor subfamily 3 group C
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Nuclear hormone receptor subfamily 3 group C member 1
Uniprot ID
P04150
Gene Name
NR3C1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000068 A-549
 Cell Line Info 
Homo sapiens (Human)  2
1
IC50 = 6.31 nM
   TI
   LI
   LO
   TS
2
IC50 = 50.12 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 12.59 nM