Brief Information of the Compound and Protein
Compound Name
 Compound Info 
2,4,6-trimethyl-N-[(2S)-1-[[6-methyl-1-(4-methylsulfonylphenyl)indazol-4-yl]amino]propan-2-yl]benzenesulfonamide
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 PubChem ID
CID: 53319310
Canonical SMILES
C[C@@H](CNc1cc(C)cc2n(ncc12)-c1ccc(cc1)S(C)(=O)=O)NS(=O)(=O)c1c(C)cc(C)cc1C
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Compound Formula C27H32N4O4S2
Compound Structure
Protein Name
 Protein Info 
Glucocorticoid receptor
Protein Classification
Transcription factor
>
Nuclear receptor
>
Nuclear hormone receptor subfamily 3
>
Nuclear hormone receptor subfamily 3 group C
>
Nuclear hormone receptor subfamily 3 group C member 1
Uniprot ID
P04150
Gene Name
NR3C1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000068 A-549
 Cell Line Info 
Homo sapiens (Human)  2
1
IC50 = 5.012 nM
   TI
   LI
   LO
   TS
2
IC50 = 12.59 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 31.62 nM