Brief Information of the Compound and Protein
Compound Name
3-((Z)-4-(((R)-2-(3,4-dimethoxyphenyl)propyl)(methyl)amino)but-2-enyl)-7,8-dimethoxy-1H-benzo[d]azepin-2(3H)-one
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PubChem ID
CID: 46937419
SID: 99445685
Canonical SMILES
COc1ccc(cc1OC)[C@@H](C)CN(C)C\C=C/CN1C=Cc2cc(OC)c(OC)cc2CC1=O
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Compound Formula C28H36N2O5
Compound Structure
Protein Name
Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 1
Protein Classification
Ion channel
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Voltage-gated ion channel
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Cyclic nucleotide-regulated channel
Uniprot ID
O88704
Gene Name
HCN1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 9410 nM
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