Brief Information of the Compound and Protein
Compound Name
N-[2-[4-(3-acetamidophenyl)piperidin-1-yl]ethyl]-1-(4-fluorophenyl)benzimidazole-2-carboxamide
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PubChem ID
CID: 49866086
Canonical SMILES
CC(=O)Nc1cccc(c1)C1CCN(CCNC(=O)c2nc3ccccc3n2-c2ccc(F)cc2)CC1
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Compound Formula C29H30FN5O2
Compound Structure
Protein Name
Melanin-concentrating hormone receptor 1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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MCH receptor
Uniprot ID
Q99705
Gene Name
MCHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  2
1
IC50 = 678 nM
   TI
   LI
   LO
   TS
2
IC50 = 973 nM
   TI
   LI
   LO
   TS