Brief Information of the Compound and Protein
Compound Name
(E)-2-cyano-N-(2,5-dimethylphenyl)-3-[1-[2-(2-furanylmethylamino)-2-oxoethyl]-3-indolyl]-2-propenamide
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PubChem ID
CID: 1140643
Canonical SMILES
Cc1ccc(C)c(NC(=O)C(=C\c2cn(CC(=O)NCc3ccco3)c3ccccc23)\C#N)c1
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Compound Formula C27H24N4O3
Compound Structure
Protein Name
Microphthalmia-associated transcription factor
Protein Classification
Transcription factor
Uniprot ID
O75030
Gene Name
MITF
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000242 SK-MEL-5 Homo sapiens (Human)  1
1
AC50 = 15211 nM
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