Brief Information of the Compound and Protein
Compound Name
(E)-N-[2-(cyclohexylamino)-2-keto-ethyl]-4-(2-hydroxy-4-methoxy-phenyl)-4-keto-N-(2-thenyl)but-2-enamide
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PubChem ID
CID: 5770968
Canonical SMILES
COc1ccc(C(=O)\C=C\C(=O)N(CC(=O)NC2CCCCC2)Cc2cccs2)c(O)c1
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Compound Formula C24H28N2O5S
Compound Structure
Protein Name
Microphthalmia-associated transcription factor
Protein Classification
Transcription factor
Uniprot ID
O75030
Gene Name
MITF
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000242 SK-MEL-5 Homo sapiens (Human)  1
1
AC50 = 20461 nM
   TI
   LI
   LO
   TS