Brief Information of the Compound and Protein
Compound Name
2-(3,4-difluorophenoxy)-N-((1s,4s)-4-(1-(4-(trifluoromethyl)phenyl)-1H-pyrrol-3-ylamino)cyclohexyl)acetamide
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Canonical SMILES
Fc1ccc(OCC(=O)N[C@H]2CC[C@H](CC2)Nc2ccn(c2)-c2ccc(cc2)C(F)(F)F)cc1F
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Compound Formula C25H24F5N3O2
Compound Structure
Protein Name
Melanin-concentrating hormone receptor 1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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MCH receptor
Uniprot ID
Q99705
Gene Name
MCHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 104 nM
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