Brief Information of the Compound and Protein
Compound Name
N-[[1-[[1-(5-tert-butylpyridin-2-yl)pyrrol-3-yl]methyl]azetidin-3-yl]methyl]-2-(3-methylphenoxy)acetamide
    Show/Hide
PubChem ID
CID: 44562524
Canonical SMILES
Cc1cccc(OCC(=O)NCC2CN(Cc3ccn(c3)-c3ccc(cn3)C(C)(C)C)C2)c1
    Show/Hide
Compound Formula C27H34N4O2
Compound Structure
Protein Name
Melanin-concentrating hormone receptor 1
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Peptide receptor (family A GPCR)
>
Short peptide receptor (family A GPCR)
>
MCH receptor
Uniprot ID
Q99705
Gene Name
MCHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 169 nM
   TI
   LI
   LO
   TS