Brief Information of the Compound and Protein
Compound Name
2-(3-chlorophenoxy)-N-(1-((1-(5-(trifluoromethyl)pyridin-2-yl)-1H-pyrrol-3-yl)methyl)piperidin-4-yl)acetamide
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PubChem ID
CID: 11554989
SID: 16657209
Canonical SMILES
FC(F)(F)c1ccc(nc1)-n1ccc(CN2CCC(CC2)NC(=O)COc2cccc(Cl)c2)c1
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Compound Formula C24H24ClF3N4O2
Compound Structure
Protein Name
Melanin-concentrating hormone receptor 1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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MCH receptor
Uniprot ID
Q99705
Gene Name
MCHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  2
1
IC50 = 48 nM
   TI
   LI
   LO
   TS
2
IC50 = 92 nM
   TI
   LI
   LO
   TS