Brief Information of the Compound and Protein
Compound Name
4-[1-(4-fluorophenyl)indazol-5-yl]-N-phenyl-N-propyl-3-(trifluoromethyl)benzenesulfonamide
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PubChem ID
CID: 46832234
SID: 99210106
Canonical SMILES
CCCN(c1ccccc1)S(=O)(=O)c1ccc(-c2ccc3n(ncc3c2)-c2ccc(F)cc2)c(c1)C(F)(F)F
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Compound Formula C29H23F4N3O2S
Compound Structure
Protein Name
Glucocorticoid receptor
Protein Classification
Transcription factor
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Nuclear receptor
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Nuclear hormone receptor subfamily 3
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Nuclear hormone receptor subfamily 3 group C
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Nuclear hormone receptor subfamily 3 group C member 1
Uniprot ID
P04150
Gene Name
NR3C1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000068 A-549 Homo sapiens (Human)  2
1
EC50 = 316.23 nM
   TI
   LI
   LO
   TS
2
IC50 = 316.23 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 15.85 nM