Brief Information of the Compound and Protein
Compound Name
 Compound Info 
2-(1-((3-(5-hydroxypyridin-2-yl)-1,2,4-oxadiazol-5-yl)methyl)cyclobutanecarboxamido)cyclohex-1-enecarboxylic acid
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 PubChem ID
CID: 135887288
SID: 93369940
Canonical SMILES
OC(=O)C1=C(CCCC1)NC(=O)C1(Cc2nc(no2)-c2ccc(O)cn2)CCC1
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Compound Formula C20H22N4O5
Compound Structure
Protein Name
 Protein Info 
Hydroxycarboxylic acid receptor 2
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Small molecule receptor (family A GPCR)
>
Carboxylic acid receptor
>
Hydroxycarboxylic acid receptor
Uniprot ID
Q8TDS4
Gene Name
HCAR2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  3
1
EC50 = 730 nM
   TI
   LI
   LO
   TS
2
Ki = 360 nM
   TI
   LI
   LO
   TS
3
Ki = 1080 nM
   TI
   LI
   LO
   TS