Brief Information of the Compound and Protein
Compound Name
N-[(1S,3R,5R)-3-Isopropyl-2-oxo-2,3-dihydrobenzoimidazole-1-carboxylic Acid(8-Azabicyclo[3.2.1]oct-3-yl)amide
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PubChem ID
SID: 85283117
Canonical SMILES
CC(C)n1c(=O)n(C(=O)N[C@H]2C[C@H]3CC[C@@H](C2)N3)c2ccccc21
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Compound Formula C18H24N4O2
Compound Structure
Protein Name
5-hydroxytryptamine receptor 4
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Serotonin receptor
Uniprot ID
Q13639
Gene Name
HTR4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  2
1
EC50 = 15.85 nM
   TI
   LI
   LO
   TS
2
Ki = 316.23 nM
   TI
   LI
   LO
   TS