Brief Information of the Compound and Protein
Compound Name
N-(2,3-dihydro-1-benzofuran-3-ylmethyl)-N-methyl-2,3,4,5-tetrahydro-1H-3-benzazepine-7-sulfonamide
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PubChem ID
CID: 42601404
SID: 74374275
Canonical SMILES
CN(CC1COc2ccccc12)S(=O)(=O)c1ccc2CCNCCc2c1
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Compound Formula C20H24N2O3S
Compound Structure
Protein Name
5-hydroxytryptamine receptor 2C
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Serotonin receptor
Uniprot ID
P28335
Gene Name
HTR2C
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  1
1
EC50 = 41 nM
   TI
   LI
   LO
   TS
CL000035 NIH 3T3 Mus musculus (Mouse)  1
1
Ki = 58 nM
   TI
   LI
   LO
   TS